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insulin receptor binding
väzba na inzulínový receptor
마지막 업데이트: 2017-04-26
사용 빈도: 1
품질:
insulin receptor binding:
väzba inzulínu na receptory:
마지막 업데이트: 2012-04-12
사용 빈도: 2
품질:
in vitro receptor binding studies have shown no measurable affinity for other than h1- receptors.
Štúdie viazania receptorov in vitro nedokázali žiadnu inú merateľnú afinitu pre iné ako h1 receptory.
마지막 업데이트: 2012-04-12
사용 빈도: 2
품질:
lurasidone also exhibits partial agonism at the 5ht-1a receptor with a binding affinity of 6.38 nm.
lurazidón prejavuje tiež čiastočný agonizmus na receptore 5ht-1a s väzbovou afinitou 6,38 nm.
마지막 업데이트: 2017-04-26
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품질:
25 dopamine, and cholinergic antagonism, consistent with the receptor-binding profile.
25 väčšiu afinitu k serotonínovým 5ht2 receptorom než k dopamínovým d2 a vyššiu 5ht2 ako d2 aktivitu na in vivo modeloch.
마지막 업데이트: 2011-10-23
사용 빈도: 1
품질:
경고: 이 정렬은 잘못되었을 수 있습니다.
잘못된 경우 삭제해 주십시오.
palonosetron is a 5-ht3 receptor antagonist with a strong binding affinity for this receptor and little or no affinity for other receptors.
palonosetrón je antagonista 5-ht3 receptora so silnou väzbovou afinitou pre tento receptor a malou alebo žiadnou afinitou k iným receptorom.
마지막 업데이트: 2017-04-26
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품질:
insulin glargine is very similar to human insulin with respect to insulin receptor binding kinetics.
vzhľadom na väzbovú kinetiku receptorov inzulínu sa inzulín glargín veľmi podobá ľudskému inzulínu.
마지막 업데이트: 2012-04-12
사용 빈도: 2
품질:
the receptor binding is long lasting due to the slow dissociation of telmisartan from the at1 receptor binding site.
väzba na receptor má dlhodobý charakter z dôvodu pomalého uvoľňovania telmisartanu z miesta väzby na receptor at1.
마지막 업데이트: 2017-04-26
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품질:
venlafaxine and odv are very similar with respect to their overall action on neurotransmitter reuptake and receptor binding.
venlafaxín a odv sú veľmi podobné vzhľadom na ich celkovú akciu na neurotransmiterové vychytávanie a receptorové viazanie.
마지막 업데이트: 2012-04-12
사용 빈도: 2
품질:
aripiprazole also exhibited moderate binding affinity for the serotonin reuptake site and no appreciable affinity for muscarinic receptors.
aripiprazol preukázal miernu afinitu aj k miestu spätného vychytávania sérotonínu a nepreukázal žiadnu afinitu k muskarínovým receptorom.
마지막 업데이트: 2017-04-26
사용 빈도: 3
품질:
aripiprazole also exhibited moderate binding affinity for the serotonin reuptake site and no appreciable affinity for cholinergic muscarinic receptors.
aripiprazol vykazoval aj stredne významnú afinitu k miestam spätného vychytávania serotonínu a žiadnu významnú afinitu k cholinergným muskarínovým receptorom.
마지막 업데이트: 2017-04-26
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품질:
the binding affinity of 4-hydroxymethyl ambrisentan for the human endothelin receptor is 65-fold less than ambrisentan.
väzbová afinita 4-hydroxymetylambrisentanu k ľudskému receptoru pre endotelín je 65-násobne nižšia ako u ambrisentanu.
마지막 업데이트: 2017-04-26
사용 빈도: 3
품질:
insulin receptor binding: in vitro studies indicate that the affinity of insulin glargine and its metabolites m1 and m2 for the human insulin receptor is similar to the one of human insulin.
väzba na inzulínový receptor: in vitro štúdie uvádzajú, že afinita inzulínu glargínu a jeho metabolitov m1 a m2 k ľudskému inzulínovému receptoru sa podobá ľudskému inzulínu.
마지막 업데이트: 2017-04-26
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품질:
in combination with its subtype selective receptor-binding characteristics, with high selectivity and low affinity for the benzodiazepine type i receptor, these properties are responsible for the overall characteristics of sonata.
v kombinácii s jeho charakteristikou subtyp-selektívnej väzby na receptor, s vysokou selektivitou a nízkou afinitou pre benzodiazepínový receptor typ i, sú tieto vlastnosti zodpovedné za celkovú charakteristiku sonaty.
마지막 업데이트: 2017-04-26
사용 빈도: 3
품질:
animal behavioural studies with olanzapine indicated 5ht, dopamine, and cholinergic antagonism, consistent with the receptor-binding profile.
behaviorálne štúdie na zvieratách preukázali antagonistické pôsobenie olanzapínu na 5ht, dopamínové a cholínergné receptory, čo je v súlade s väzbovým profilom látky.
마지막 업데이트: 2017-04-26
사용 빈도: 3
품질:
animal behavioral studies with 1 olanzapine indicated 5ht, dopamine, and cholinergic antagonism, consistent with the receptor- binding profile.
s inými centrálne pôsobiacimi liekmi čalkoholom.
마지막 업데이트: 2011-10-23
사용 빈도: 1
품질:
경고: 이 정렬은 잘못되었을 수 있습니다.
잘못된 경우 삭제해 주십시오.
the binding affinity of 99mtc-depreotide to sstr was shown in studies of pancreatic tumours in lewis rats and in vitro in human tumour membranes.
väzbová afinita 99mtc-depreotidu na sstr bola dokázaná v štúdiách nádorov pankreasu u potkanov lewis a in vitro u ľudských nádorových membrán.
마지막 업데이트: 2017-04-26
사용 빈도: 3
품질:
the binding affinity (ki) of eluxadoline for human κor has not been determined; however, the ki for guinea pig cerebellum κor is 55 nm.
väzobná afinita (ki) eluxadolínu k ľudským κor nebola stanovená, avšak hodnota ki pre κor v cerebelle morčiat je 55 nm.
마지막 업데이트: 2017-04-26
사용 빈도: 1
품질:
for toremifene, which has a relatively high binding affinity for sugammadex and for which relatively high plasma concentrations might be present, some displacement of vecuronium or rocuronium from the complex with sugammadex could occur.
pri toremifene, ktorý má relatívne vysokú väzbovú afinitu k sugammadexu a ktorý môže dosiahnuť relatívne vysoké plazmatické koncentrácie, sa môže objaviť vytesnenie vekurónia alebo rokurónia z komplexu so sugammadexom.
마지막 업데이트: 2017-04-26
사용 빈도: 1
품질:
cellular uptake does not require receptors, binding proteins or metabolic processes and does not occur by pinocytosis.
prienik do buniek si nevyžaduje receptory, väzbové proteíny alebo metabolické procesy a neuskutočňuje sa pinocytózou.
마지막 업데이트: 2017-04-26
사용 빈도: 1
품질: