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cependant ces dérivés de perhydroisoindolone ne manifestent pas d'activité antagoniste des récepteurs nk2.
however, these perhydroisoindolone derivatives do not display any antagonistic activity to nk2 receptors.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite:
on obtient 48,7 g de chlorhydrate de bis(fluoro-3 phényl)-7,7 perhydroisoindolone-4.
7,7-bis(3-fluorophenyl)perhydro-4-isoindolone hydrochloride (48.7 g) is obtained.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite:
on obtient 6,4 g de d-mandélate de diphényl-7,7 perhydroisoindolone-4-(3as,7as).
6.4 g of (3as,7as)-7,7-diphenyl-perhydroisoindol-4-one d-mandelate are obtained.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite:
la préparation du dérivé de la perhydroisoindolone de formule générale (v) s'effectue par analogie avec la méthode décrite dans la demande de brevet européen ep 429 366.
the preparation of the perhydroisoindolone derivative of the general formula (v) is carried out by a method analogous to that described in european patent application ep 429 366.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite:
on obtient 13 g de diphényl-7,7 perhydroisoindolone-4-(3ars,7ars) sous forme d'une meringue blanche.
(3ars,7ars)-7,7-diphenyl-4-perhydroisoindolone (13 g) is obtained in the form of a white meringue.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite:
le dérivé de perhydroisoindolone de formule générale (viii) peut être préparé comme décrit ci-après dans les exemples et par analogie avec les méthodes décrites dans la demande de brevet ep 429 366.
the perhydroisoindolone derivative of general formula (viii) can be prepared as described below in the examples and by analogy with the methods described in the patent application ep 429 366.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite:
a partir des fractions 9 à 15 réunies et concentrées à sec sous pression réduite (2,7 kpa) , on obtient 31 g de allyloxycarbonyl-7 benzyl-2 méthyl-7 perhydroisoindolone-4-(3ars,7sr,7ars) sous forme d'huile.
from fractions 9 to 15, which are combined and concentrated to dryness under reduced pressure (2.7 kpa), 31 g of (3ars,7sr,7ars)-7-allyloxycarbonyl2-benzyl-7-methyl-4-perhydroisoindolone are obtained in oil form.
Son Güncelleme: 2014-12-03
Kullanım Sıklığı: 1
Kalite: