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lurasidone does not bind to histaminergic or muscarinic receptors.
lurasidon se ne veže na histaminergične ali muskarinske receptorje.
Last Update: 2017-04-26
Usage Frequency: 1
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it weakly inhibits dopamine reuptake with no significant affinity for histaminergic, dopaminergic, cholinergic and adrenergic receptors.
Šibko zavira prevzem dopamina brez pomembne afinitete za histaminergične, dopaminergične, holinergične in adrenergične receptorje.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
venlafaxine has virtually no affinity for rat brain muscarinic, cholinergic, h1-histaminergic or α 1-adrenergic receptors in vitro.
25 venlafaksin v podganjih možganih in vitro praktično nima afinitete za muskarinske, holinergične, h1- histaminske ali α1- adrenergične receptorje.
Last Update: 2012-04-11
Usage Frequency: 4
Quality:
binding studies indicate that agomelatine has no effect on monoamine uptake and no affinity for , adrenergic, histaminergic, cholinergic, dopaminergic and benzodiazepine receptors.
Študije o vezavi so pokazale, da agomelatin nima učinka na privzem monoaminov niti afinitete za α-adrenergične, β-adrenergične, histaminske, holinergične, dopaminergične ali benzodiazepinske receptorje.
Last Update: 2017-04-26
Usage Frequency: 1
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paliperidone also blocks alfa1-adrenergic receptors and blocks, to a lesser extent, h1-histaminergic and alfa2-adrenergic receptors.
paliperidon zavira tudi adrenergične receptorje alfa-1 in v manjši meri, tudi histaminske receptorje h1 in adrenergične receptorje alfa-2.
Last Update: 2017-04-26
Usage Frequency: 7
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risperidone binds also to alpha1-adrenergic receptors, and, with lower affinity, to h1-histaminergic and alpha2-adrenergic receptors.
risperidon se prav tako veže na α1 - adrenergične receptorje in z manjšo afiniteto na histaminske h1 in α 2- adrenergične receptorje.
Last Update: 2012-04-11
Usage Frequency: 2
Quality:
pitolisant is a potent, orally active histamine h3-receptor antagonist/inverse agonist which, via its blockade of histamine auto-receptors enhances the activity of brain histaminergic neurons, a major arousal system with widespread projections to the whole brain.
pitolizant je močan, peroralno aktiven antagonist/inverzni agonist histaminskih receptorjev h3, ki z zaviranjem histaminskih avtoreceptorjev spodbuja aktivnost histaminergičnih nevronov v možganih, pomembnega sistema, ki skrbi za budnost in katerega projekcije segajo v vse predele možganov.
Last Update: 2017-04-26
Usage Frequency: 1
Quality: