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telziri toimeaine fosamprenaviir on eelravim, mis muundub organismis proteaasiinhibiitoriks amprenaviiriks.
the active substance in telzir, fosamprenavir, is a ‘prodrug’ of the protease inhibitor amprenavir, which means that it is converted into amprenavir in the body.
prasugreel on eelravim ja metaboliseerub in vivo kiiresti aktiivseks metaboliidiks ja inaktiivseteks metaboliitideks.
prasugrel is a prodrug and is rapidly metabolised in vivo to an active metabolite and inactive metabolites.
tenofoviirdisoproksiilfumaraat on vesilahustuv ester, eelravim, mis muudetakse in vivo kiiresti tenofoviiriks ja formaldehüüdiks.
tenofovir disoproxil fumarate is a water soluble ester prodrug which is rapidly converted in vivo to tenofovir and formaldehyde.
indoksakarb on eelravim, mille farmakodünaamiliste toimete avaldumiseks on vajalik bioaktiviseerumine ainele tundlike putukate ensüümide abil.
indoxacarb is a pro- drug that requires bioactivation by enzymes in susceptible insects to exert its pharmacodynamic effects.