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rivastigminas blokuoja acetilcholin skaidanci ferment acetilcholinesterazs ir butirilcholinesterazs veikl.
rivastigmine works by blocking the enzymes which break down acetylcholine: acetylcholinesterase and butyrylcholinesterase.
最后更新: 2008-03-04
使用频率: 2
质量:
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rivastigminas yra karbamato tipo acetilcholinesterazs ir butirilcholinesterazs inhibitorius, pagerinantis cholinerginio impulso perdavim neuronais, neleisdamas skaidyti sveik neuron isskirt acetilcholin.
rivastigmine is an acetyl-and butyrylcholinesterase inhibitor of the carbamate type, thought to facilitate cholinergic neurotransmission by slowing the degradation of acetylcholine released by functionally intact cholinergic neurones.
最后更新: 2008-03-04
使用频率: 10
质量:
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rivastigminas yra karbamato tipo acetilcholinesterazs ir butirilcholinesterazs inhibitorius, pagerinantis cholinerginio impulso perdavim neuronais, neleisdamas skaidyti sveik cholinergini neuron isskirt acetilcholin.
rivastigmine is an acetyl-and butyrylcholinesterase inhibitor of the carbamate type, thought to facilitate cholinergic neurotransmission by slowing the degradation of acetylcholine released by functionally intact cholinergic neurones.
最后更新: 2008-03-04
使用频率: 4
质量:
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rivastigmino pusins eliminacijos periodas yra apie 1 val., o acetilcholinesterazs inhibicija trunka mazdaug 9 valandas, todl, jei perdozavimas kliniskai nepasireiskia, rekomenduojama 24 valandas
as rivastigmine has a plasma half-life of about 1 hour and a duration of acetylcholinesterase inhibition of about 9 hours, it is recommended that in cases of asymptomatic overdose no further dose of rivastigmine should be administered for the next 24 hours.
最后更新: 2008-03-04
使用频率: 2
质量:
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rivastigmino pusins eliminacijos periodas yra apie 1 val., o acetilcholinesterazs inhibicija trunka mazdaug 9 valandas, todl, jei perdozavimas kliniskai nepasireiskia, rekomenduojama 24 valandas nevartoti rivastigmino.
as rivastigmine has a plasma half-life of about 1 hour and a duration of acetylcholinesterase inhibition of about 9 hours, it is recommended that in cases of asymptomatic overdose no further dose of rivastigmine should be administered for the next 24 hours.
最后更新: 2008-03-04
使用频率: 8
质量:
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sveikiems jauniems vyrams geriamoji 3 mg vaisto doz apie 40% sumazina acetilcholinesterazs (ache) aktyvum likvore per pirmsias 1, 5 valandas po vartojimo.
in healthy young men, an oral 3 mg dose decreases acetylcholinesterase (ache) activity in csf by approximately 40% within the first 1.5 hours after administration.
最后更新: 2008-03-04
使用频率: 14
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in vitro nustatyta, kad sis metabolitas labai silpnai slopina acetilcholinesteraz ( 10%) .
in vitro, this metabolite shows minimal inhibition of acetylcholinesterase ( 10%) .
最后更新: 2008-03-04
使用频率: 14
质量:
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