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sekä vardenafiilin että m1:n proteiiniinsitoutuminen on riippumatonta lääkkeen kokonaispitoisuudesta.
for vardenafil as well as m1, protein binding is independent of total drug concentrations.
Last Update: 2017-04-26
Usage Frequency: 9
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päämetaboliitin (parahydroksisulfaatti) proteiiniinsitoutuminen on hyvin voimakasta (> 99, 99%).
the protein binding of the major metabolite (a para-hydroxy-sulphate) is very high (> 99.99%).
Last Update: 2012-04-10
Usage Frequency: 6
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päämetaboliitin (parahydroksisulfaatti) proteiiniinsitoutuminen on hyvin voimakasta ( 99,99 %).
the protein binding of the major metabolite (a para-hydroxy-sulphate) is very high (> 99.99%).
Last Update: 2017-04-26
Usage Frequency: 1
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vakaassa tilassa lopinaviirin proteiiniinsitoutuminen pysyy vakiona mittausalueella, joka saavutetaan antamalla 400/100 mg kaletraa kahdesti päivässä, ja se on samankaltainen terveillä ja hiv-positiivisilla potilailla.
at steady state, lopinavir protein binding remains constant over the range of observed concentrations after 400/100 mg kaletra twice daily, and is similar between healthy volunteers and hiv-positive patients.
Last Update: 2008-03-04
Usage Frequency: 3
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in vitro -tutkimukset osoittavat, että ertapeneemin vaikutus voimakkaasti proteiiniin sitoutuvien lääkevalmisteiden (varfariini, etinyyliestradioli ja noretisteroni) proteiiniinsitoutumiseen plasmassa on pieni.
in-vitro studies indicate that the effect of ertapenem on the plasma protein binding of highly protein bound medicinal products (warfarin, ethinyl estradiol, and norethindrone) was small.
Last Update: 2017-04-26
Usage Frequency: 4
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